Table 3. k2/Ks second order rate constants for acylation.
PBP2 Variant | k2/KS (M−1s−1) | ||
---|---|---|---|
Cefixime | Ceftriaxone | Penicillin G | |
PBP2 | 1480000 ± 22000 | 1710000 ± 90000 | 75700 ± 2300 |
PBP235/02 | 7170 ± 280 | 11300 ± 440 | 510 ± 90 |
PBP235/02-A501T | 5550 ± 160 | 30400 ± 300 | 1860 ± 130 |
PBP235/02-A501V | 3150 ± 120 | 20000 ± 390 | 1370 ± 140 |
PBP235/02-A501R | 820 ± 40 | 6460 ± 70 | 960 ± 100 |
PBP235/02-A501P | 40 ± 1 | 250 ± 20 | 810 ± 40 |