. 2017 Jun 1;8(7):737–741. doi: 10.1021/acsmedchemlett.7b00132

Table 1. SAR for N-Alkyl Substitutions Extending from the Piperidine^a.

All bromodomain assays were run in TR-FRET format. IC₅₀ data are an average of at least two independent experiments. Assay tables with standard deviations are located in the Supporting Information. A full table of data with standard deviations for these and other N-alkyl substituents can be found in the Supporting Information.

Table 1. SAR for N-Alkyl Substitutions Extending from the Piperidinea.

Table 1. SAR for N-Alkyl Substitutions Extending from the Piperidine^a.