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. Author manuscript; available in PMC: 2018 Jul 15.
Published in final edited form as: Neuropharmacology. 2017 Apr 27;121:167–178. doi: 10.1016/j.neuropharm.2017.04.038

Table 1.

GABA sensitivity of different GABAA receptor configurations

Receptor configurations EC50 (μM) Hill coefficient Sample size EC30 (μM)
α1β2γ 2 34 ± 4.9 1.08 ± 0.15 8 10
α2β2γ2 40 ± 2.3 1.48 ± 0.11 6 23
α3β2γ21 33 ± 2.1 1.1 ± 0.03 4 20
α4β2γ2 4.3 ± 0.2 1.19 ±0.05 5 2
α5β2γ2 16 ± 1.0 1.27 ± 0.09 4 9
α6β2γ21 1.6 ± 0.1 1.6 ± 0.11 4 1
α1β22 1.6 ± 0.2 1.3 ± 0.10 4 0.5
α1(T6′F)β22 1.7 ± 0.3 0.9 ± 0.10 4 0.5
α1β2(T6′F)2 3.6 ± 0.5 1.1 ± 0.10 4 1.2
α1(R84P)β2γ2 7.9 ± 1.2 1.54 ± 0.21 7 4
α1(M89L)β2γ2 6.6 ± 0.5 1.50 ± 0.08 4 4
α1(I120L)β2γ2 32 ± 1.0 1.17 ±0.04 5 10
α1(R84P/M89L)β2γ2 4.1 ± 0.1 0.93 ± 0.03 5 1.7
α1(R84P/M89L/I120L)β2γ2 5.3 ± 0.4 1.24 ± 0.09 4 2.5

1, 2. indicate the values reported in our previous publications: