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. Author manuscript; available in PMC: 2018 Apr 7.
Published in final edited form as: J Am Chem Soc. 2016 Oct 13;138(42):14092–14099. doi: 10.1021/jacs.6b08942

Table 3.

Scope of the aminesa,b

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a

Reaction conditions: 1a (35.6 mg, 0.1 mmol), Aminating reagent (1.5 equiv.), Pd(OAc)2 (15 mol%), L28 (15 mol%), NBE-CO2Me (42.8 mg, 3 equiv.), AgOAc (50.1 mg, 3.0 equiv.), CH2Cl2 (1.0 mL), 100 °C, Air, 24 h.

b

Isolated yield.

c

Pd(OAc)2 (10 mol%), L28 (10 mol%), NBE-CO2Me (21.4 mg, 1.5 equiv.), AgOAc (33.4 mg, 2.0 equiv.) were used.