Table 2.
Operational analysis with bias factors (ΔΔLogR ± error) comparing Gαi (no PTX) with Gαs (with PTX) signalling of moderate expression 3HA‐hCB1 HEK cells
CP55,940 | WIN55,212‐2 | AEA | 2‐AGa | THC | BAY | |
---|---|---|---|---|---|---|
ΔΔLogR | 0.29 ± 0.37 | 0.19 ± 0.29 | 0.53 ± 0.27 | 0.00 ± 0.29 | NDb | NDb |
2‐AG was used as the reference ligand.
As no Gαs signal was observed for THC or BAY, a bias factor could not be determined.