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. Author manuscript; available in PMC: 2017 Aug 26.
Published in final edited form as: Angew Chem Int Ed Engl. 2016 Aug 1;55(36):10578–10599. doi: 10.1002/anie.201600791

Table 5.

Rh(III)-catalyzed C(sp2)–H annulation with α-(pseudo)halo ketones using the N-methoxy amide directing group (Glorius et al., 2014).[73]

graphic file with name nihms877172u6.jpg
Entry X % Yield[a]
1 X = Br 10[b]
2 X = Cl 62
3 X = OTs 86
4 X = OMs 86
5 X = OBz 0
[a]

Isolated yield.

[b]

1H NMR yield.