Table 1.
EC50 values (from n = 3 experiments) for AIP-I and its derivatives and IC50 values (from n = 4 experiments) for TrAIP-II and its derivatives when AIP-I is present at 100 nM (i.e., the EC95).
EC50 (nM) | AIP-I | 28 (± 3) |
Alkyne-AIP-I | 190 (± 40) | |
PEG330-triazole-AIP-I | 1100 (± 200) | |
IC50 (μM) | TrAIP-II | 1.5 (± 0.5) |
Alkyne-TrAIP-II | 0.21 (± 0.05) | |
PEG330-triazole-TrAIP-II | 3.1 (± 1.5) |