Table 3.
| ||||
---|---|---|---|---|
entry | indole | product | % yield 2 | % yield 3 |
1 |
1b |
2i |
66% | 5% |
2 |
1c |
2j |
47% | 9% |
3 |
1d |
2k |
51% | 10% |
4 |
1e |
2l |
70% | 10% |
5 |
1f |
2m |
64% | 14% |
6 |
1g |
2n |
61% | 17% |
Conditions: 2 equiv indole, 1 equiv PhI, 4 equiv KOtBu