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. Author manuscript; available in PMC: 2017 Aug 4.
Published in final edited form as: Angew Chem Int Ed Engl. 2017 Mar 3;56(14):3951–3955. doi: 10.1002/anie.201612311

Table 3.

Scope of Indole

graphic file with name nihms882669u3.jpg
entry indole product % yield 2 % yield 3
1 graphic file with name nihms882669t21.jpg
1b
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2i
66% 5%
2 graphic file with name nihms882669t23.jpg
1c
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2j
47% 9%
3 graphic file with name nihms882669t25.jpg
1d
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2k
51% 10%
4 graphic file with name nihms882669t27.jpg
1e
graphic file with name nihms882669t28.jpg
2l
70% 10%
5 graphic file with name nihms882669t29.jpg
1f
graphic file with name nihms882669t30.jpg
2m
64% 14%
6 graphic file with name nihms882669t31.jpg
1g
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2n
61% 17%

Conditions: 2 equiv indole, 1 equiv PhI, 4 equiv KOtBu