Skip to main content
. Author manuscript; available in PMC: 2018 May 9.
Published in final edited form as: ChemMedChem. 2017 Apr 18;12(9):660–677. doi: 10.1002/cmdc.201600636

Figure 2.

Figure 2

Concentration-dependent study for 1 and one of its analogs, 6, using a radiometric assay at Reaction Biology Corp showed that the compounds inhibited enzyme activity by an IC50 of about 5 μM.