Table 2. Development of HDL-mimicking α-tocopherol-coated NPs. Listed are the compositions per 1 ml NPs.
(A) The array #1 with high contents of CO without TPGS, (B) modified 2 A by adding TPGS into the compositions, (C) The array #2 with low contents of CO without TPGS, and (D) modified 2C by adding TPGS into the composition.
| A.
| ||||||
|---|---|---|---|---|---|---|
| Experiment | PC (µg) | SM (µg) | PS (µg) | CO (µg) | Particle size (nm) | P.I. |
| 1–1 | 32 | 6 | 4 | 40 | 275.4 | 0.265 |
| 1–2 | 32 | 6 | 4 | 50 | 383.4 | 0.181 |
| 1–3 | 32 | 6 | 4 | 60 | 242.9 | 0.295 |
| 1–4 | 40 | 7.5 | 5 | 40 | 284.1 | 0.31 |
| 1–5 | 40 | 7.5 | 5 | 50 | 333.6 | 0.301 |
| 1–6 | 40 | 7.5 | 5 | 60 | 404.1 | 0.193 |
| 1–7 | 48 | 9 | 6 | 40 | 386.4 | 0.284 |
| 1–8 | 48 | 9 | 6 | 50 | 282.6 | 0.297 |
| 1–9 | 48 | 9 | 6 | 60 | 255.2 | 0.255 |
| B.
| |||||||
|---|---|---|---|---|---|---|---|
| Experiment | PC (µg) | SM (µg) | PS (µg) | CO (µg) | TPGS (µg) | Particle size (nm) | P.I. |
| 2–1 | 32 | 6 | 4 | 40 | 60 | 173 | 0.261 |
| 2–2 | 32 | 6 | 4 | 50 | 40 | 181.9 | 0.236 |
| 2–3 | 32 | 6 | 4 | 60 | 20 | 198.7 | 0.223 |
| 2–4 | 40 | 7.5 | 5 | 40 | 30 | 173.1 | 0.263 |
| 2–5 | 40 | 7.5 | 5 | 50 | 40 | 190 | 0.239 |
| 2–6 | 40 | 7.5 | 5 | 60 | 20 | 166 | 0.27 |
| 2–7 | 48 | 9 | 6 | 40 | 30 | 173.1 | 0.271 |
| 2–8 | 48 | 9 | 6 | 50 | 10 | 202 | 0.28 |
| 2–9 | 48 | 9 | 6 | 60 | 20 | 211.4 | 0.294 |
| C.
| ||||||
|---|---|---|---|---|---|---|
| Experiment | PC (µg) | SM (µg) | PS (µg) | CO (µg) | Particle size (nm) | P.I. |
| 3–1 | 40 | 7.5 | 2.5 | 5 | 246.6 | 0.312 |
| 3–2 | 40 | 7.5 | 2.5 | 10 | 301.7 | 0.307 |
| 3–3 | 56 | 10.5 | 3.5 | 5 | 269.2 | 0.234 |
| 3–4 | 56 | 10.5 | 3.5 | 10 | 296.1 | 0.332 |
| D.
| |||||||
|---|---|---|---|---|---|---|---|
| Experiment | PC (µg) | SM (µg) | PS (µg) | CO (µg) | TPGS (µg) | Particle size (nm) | P.I. |
| 4–1 | 40 | 7.5 | 2.5 | 5 | 30 | 192.7 | 0.259 |
| 4–2 | 40 | 7.5 | 2.5 | 10 | 30 | 178.9 | 0.283 |
| 4–3 | 56 | 10.5 | 3.5 | 5 | 50 | 171.6 | 0.295 |
| 4–4 | 56 | 10.5 | 3.5 | 10 | 50 | 162 | 0.268 |