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. 2017 Jul 6;8(32):52026–52044. doi: 10.18632/oncotarget.19036

Table 1B. IC50s (nM) (mean+/−S.D.), generated using GraphPad Prism 7 Software, for crenolanib and AC220 tested against Ba/F3-FLT3-ITD and Ba/F3-FLT3-ITD+SYK-TEL. Cell growth assays were carried out for approximately 3 days.

crenolanib
(IC50, nM)
quizartinib
(IC50, nM)
Ba/F3-FLT3-ITD 6.2+/−2 0.3+/−0.3
Ba/F3-FLT3-ITD+SYK-TEL 520.6+/−121.1 627.5+/−32.2