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. Author manuscript; available in PMC: 2018 Jun 1.
Published in final edited form as: Clin Cancer Res. 2016 Nov 23;23(11):2869–2879. doi: 10.1158/1078-0432.CCR-16-1742

Scheme I.

Scheme I

a) Pd(II)acetate, BINAP, K3PO4, dioxane, 100 °C, 17 h; b) 4N HCl in dioxane; c) Pd(II)acetate, BINAP, K3PO4, dioxane, 100 °C, 15 h; d) Methanol, 4N HCl in dioxane