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. Author manuscript; available in PMC: 2018 Feb 1.
Published in final edited form as: Bioorg Med Chem. 2016 Nov 30;25(3):864–869. doi: 10.1016/j.bmc.2016.11.056

Table 5.

Antibacterial activity against S. aureus clinical strains

Compd MIC (µM)
USA200 USA300 USA400 UAMS-1 Newman Mu50
3e 6.2 6.2 6.2 25 6.2 6.2
3d <1.5 3.1 3.1 12.5–25 3.1 3.1
5 25 12.5–25 12.5 >=25 12.5 25
3i 6.2 6.2 6.2 12.5 6.2 6.2
3k 12.5 12.5 12.5 >25 12.5 >25
3l 3.1 12.5 3.1 6.2 3.1–6.2 6.2
Daptomycin1 0.78 0.78 0.78 >12.5 ND2 3.1
1

Taken from ref. 19.

2

Not determined.