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. 2017 Jun 28;8(38):63187–63207. doi: 10.18632/oncotarget.18730

Table 2. H3K9Me2 cell immunofluorescence In-Cell Western (ICW) assay results (MDA-MB-231 cell line).

Compound G9a IC50 (μM) Compound G9a IC50 (μM)
4 96.69±1.68 4a 74.21±1.94
5 >100 5a 66.63±3.98
6 >100 6a >100
7 76.74±0.89 7a 54.55±3.05
13 37.79±2.80 13a >100
14 7.136±1.62 14a 46.83±1.97
15 72.10±1.37 15a 46.97±3.33
16 90.26±3.75 16a 45.71±1.76
19 99.63±3.13 21 ND
20 97.51±2.78 22 60.65±3.66
BIX-01294 4.563±1.2 5b 87.39±5.44