Table 47.
ABP | IC50, nM | |||||
---|---|---|---|---|---|---|
| ||||||
Casp-3 | Casp-6 | Casp-7 | Casp-8 | Casp-9 | ||
FAM-DEVD-AOMK | 540 | 18 | 26 | 24 | 29 | 1100 |
FAM-CV3-AOMK | 541 | 27 | 3000 | 1300 | 100 | 3100 |
Biotin-DEVD-AOMK | 542 | 39 | 75 | 38 | 50 | 1100 |
Biotin-CV3-AOMK | 543 | 13 | 1200 | 420 | 53 | 2500 |
Rho-Ahx2-DW3-KE | 544 | 25 | 4000 | 3500 | 930 | ND |
Rho-DEVD-AOMK | 545 | 10 | 65 | 17 | 12 | ND |
Biotin-CV8/9-KE | 546 | 4500 | ND | ND | 170 | ND |