Table 2. Bis(imino)pyridine Substituent Effects on the Time to Reach >98% Conversion in the [2π + 2π] Cycloaddition of N,N-Diallyl-4-fluoroaniline.
entry | [Co] | time (h)a |
---|---|---|
1 | (iPrPDI)CoN2 (1) | 8 |
2 | (TricPDI)CoN2 (2) | 1 |
3 | (EtPDI)CoN2 (3) | 44 |
4 | (MePDI)CoN2 (4) | 60 |
5 | (iPrEtPDI)CoN2 (5) | >72b |
6 | (iPriPrPDI)CoN2 (6) | >72c |
7 | 4-pyrr-(iPrPDI)CoN2 (7) | 36d |
Time to >98% conversion.
41% conversion at 72 h.
7% conversion at 72 h.
48% cycloaddition and 52% alkene isomerization products.