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. 2017 Sep 7;8(10):1093–1098. doi: 10.1021/acsmedchemlett.7b00296

Table 1. SAR of 4,6-Disubstituted Indazoles.

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*

Data is mean of at least three separate test occasions unless stated.

a

Data from in-house PIM1 assay, n = 1.

b

Tested <4.6 on one occasion.

c

Data from in-house PIM1 assay.

d

Tested <4.6 on two occasions.

e

Tested <4.6 on three occasions.

f

GSK3β data was generated at Reaction Biology Corporation.23

g

Tested <4.6 on four occasions.

h

n = 1.

i

n = 2.