Nomenclature | bromodomain adjacent to zinc finger domain 2A | bromodomain adjacent to zinc finger domain 2B | CREB binding protein | polybromo 1 | SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a, member 4 |
HGNC, UniProt | BAZ2A, Q9UIF9 | BAZ2B, Q9UIF8 | CREBBP, Q92793 | PBRM1, Q86U86 | SMARCA4, P51532 |
Selective inhibitors | GSK2801 (pK d 6.6) [73] | GSK2801 (pK d 6.9) [73] | I‐CBP112 (pK d 6.8) [72] | PFI‐3 (pK d 7.3) [79] | PFI‐3 (pK d 7.1) [79] |