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. 2017 Oct 21;174(Suppl Suppl 1):S272–S359. doi: 10.1111/bph.13877
Nomenclature BMX non‐receptor tyrosine kinase Bruton tyrosine kinase TXK tyrosine kinase
HGNC, UniProt BMX, P51813 BTK, Q06187 TXK, P42681
EC number 2.7.10.2 2.7.10.2 2.7.10.2
Common abreviation Etk Btk TXK
Inhibitors compound 38 (pIC50 9.1) [300], ibrutinib (pIC50 9.1) [318], compound 31 (pIC50 8.7) [300] ibrutinib (pIC50 9.3) [395], compound 31 (pIC50 8.4) [300], compound 38 (pIC50>8.4) [300]
Selective inhibitors BMX‐IN‐1 (pIC50 8.1) [307] CGI1746 (pIC50 8.7) [120], CHMFL‐BTK‐11 (Irreversible inhibition) (pIC50 7.6) [576]