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. 2017 Oct 21;174(Suppl Suppl 1):S17–S129. doi: 10.1111/bph.13878
Nomenclature TA 1 receptor
HGNC, UniProt TAAR1, Q96RJ0
Potency order of endogenous ligands tyramine>β ‐phenylethylamine>octopamine = dopamine [189]
Agonists RO5166017 [1648]
Antagonists EPPTB (Inverse agonist) (pIC50 5.1) [205]
Labelled ligands [3 H]tyramine (Agonist) [189]