| Nomenclature | 5‐HT 1D receptor | 5‐ht 1e receptor | 5‐HT 1F receptor |
| HGNC, UniProt | HTR1D, P28221 | HTR1E, P28566 | HTR1F, P30939 |
| Agonists | dihydroergotamine [719, 1150, 1157], ergotamine [648], L‐694,247 [2140], naratriptan [457, 1425, 1651], zolmitriptan [1425], frovatriptan [2158], rizatriptan [1425] | BRL‐54443 [232] | BRL‐54443 [232], eletriptan [1425], sumatriptan [12, 13, 1425, 2052] |
| Selective agonists | PNU109291 [511] – Gorilla, eletriptan [1425] | – | lasmiditan [1439], LY334370 [2052], 5‐BODMT [1014], LY344864 [1572] |
| Selective antagonists | SB 714786 (pK i 9.1) [2074] | – | – |
| Labelled ligands | [3 H]eletriptan (Agonist) [1425], [3 H]alniditan (Agonist) [1150], [125 I]GTI (Selective Agonist) [197, 237] – Rat, [3 H]GR 125,743 (Selective Antagonist) (pK d 8.6) [2150], [3 H]sumatriptan (Agonist) [1425] | [3 H]5‐HT (Agonist) [1299, 1532] | [3 H]LY334370 (Agonist) [2052], [125 I]LSD (Agonist) [45] – Mouse |
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