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. 2017 Oct 21;174(Suppl Suppl 1):S17–S129. doi: 10.1111/bph.13878

Nomenclature	GPER
HGNC, UniProt	GPER1, Q99527
Agonists	raloxifene [1570]
Selective agonists	G1 [179]
Selective antagonists	G36 (pIC₅₀ 6.8–6.9) [438], G15 (pIC₅₀ 6.7) [437]
Labelled ligands	[³ H]17 β‐estradiol (Agonist) [1953]