| Nomenclature | GLP‐2 receptor | glucagon receptor | secretin receptor |
| HGNC, UniProt | GLP2R, O95838 | GCGR, P47871 | SCTR, P47872 |
| Endogenous agonists | glucagon‐like peptide 2 (GCG, P01275) [1958] | glucagon (GCG, P01275) [1587] | secretin (SCT, P09683) [343] |
| Agonists | teduglutide [1310] | – | – |
| Selective antagonists | – | L‐168,049 (pIC50 8.4) [282], adomeglivant (pK i 8.2) [963, 967], des‐His 1‐[Glu9]glucagon‐NH2 (pA2 7.2) [2004, 2005] – Rat, NNC 92‐1687 (pK i 5) [1234], BAY27‐9955 [1566] | [(CH 2NH)4,5]secretin (pK i 5.3) [704] |
| Labelled ligands | – | [125 I]glucagon (human, mouse, rat) (Agonist) | [125 I](Tyr 10)secretin‐27 (rat) (Agonist) [2001] – Rat |
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