Nomenclature | kisspeptin receptor |
HGNC, UniProt | KISS1R, Q969F8 |
Endogenous agonists | kisspeptin‐10 (KISS1) [1041, 1501], kisspeptin‐54 (KISS1, Q15726) [1041, 1501], kisspeptin‐14 (KISS1, Q15726) [1041], kisspeptin‐13 (KISS1, Q15726) [1041] |
Selective agonists | 4‐fluorobenzoyl‐FGLRW‐NH2 [1973], [dY]1 KP‐10 [401] – Mouse |
Selective antagonists | peptide 234 [1674] |
Labelled ligands | [125I]Tyr45 ‐kisspeptin‐15 (Agonist) [1501], [125 I]kisspeptin‐13 (human) (Agonist) [1314], [125 I]kisspeptin‐10 (human) (Agonist) [1041], [125 I]kisspeptin‐14 (human) (Agonist) [1314] |