Skip to main content
. 2017 Oct 21;174(Suppl Suppl 1):S17–S129. doi: 10.1111/bph.13878
Nomenclature kisspeptin receptor
HGNC, UniProt KISS1R, Q969F8
Endogenous agonists kisspeptin‐10 (KISS1) [1041, 1501], kisspeptin‐54 (KISS1, Q15726) [1041, 1501], kisspeptin‐14 (KISS1, Q15726) [1041], kisspeptin‐13 (KISS1, Q15726) [1041]
Selective agonists 4‐fluorobenzoyl‐FGLRW‐NH2 [1973], [dY]1 KP‐10 [401] – Mouse
Selective antagonists peptide 234 [1674]
Labelled ligands [125I]Tyr45 ‐kisspeptin‐15 (Agonist) [1501], [125 I]kisspeptin‐13 (human) (Agonist) [1314], [125 I]kisspeptin‐10 (human) (Agonist) [1041], [125 I]kisspeptin‐14 (human) (Agonist) [1314]