Nomenclature | NTS 1 receptor | NTS 2 receptor |
HGNC, UniProt | NTSR1, P30989 | NTSR2, O95665 |
Potency order of endogenous ligands | neurotensin (NTS, P30990) >neuromedin N {Mouse, Rat} [776] | neurotensin (NTS, P30990) = neuromedin N {Mouse, Rat} [1297] |
Selective agonists | JMV449 [1822] – Rat | levocabastine [1297, 1657] |
Selective antagonists | meclinertant (pIC50 7.5–8.2) [699] | – |
Labelled ligands | [3 H]meclinertant (Antagonist) (pK d 8.5) [1085] – Rat | – |