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. 2017 Oct 21;174(Suppl Suppl 1):S17–S129. doi: 10.1111/bph.13878
Nomenclature NTS 1 receptor NTS 2 receptor
HGNC, UniProt NTSR1, P30989 NTSR2, O95665
Potency order of endogenous ligands neurotensin (NTS, P30990) >neuromedin N {Mouse, Rat} [776] neurotensin (NTS, P30990) = neuromedin N {Mouse, Rat} [1297]
Selective agonists JMV449 [1822] – Rat levocabastine [1297, 1657]
Selective antagonists meclinertant (pIC50 7.5–8.2) [699]
Labelled ligands [3 H]meclinertant (Antagonist) (pK d 8.5) [1085] – Rat