Table 2.
Site specificity of anti-Aβ antibody in patients by peptide epitope mapping
Peptide sequence | Aβ position | Subjects |
||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
P101 | P102 | P103 | P104 | P105 | P106 | P107 | P108 | P109 | P201 | P202 | P203 | P204 | P205 | P206 | P207 | P208 | P209 | P210 | ||
TEEISEVKMD | −9 to 1 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
EEISEVKMDA | −8 to 2 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
EISEVKMDAE | −7 to 3 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
ISEVKMDAEF | −6 to 4 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
SEVKMDAEFR | −5 to 5 | 10 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
EVKMDAEFRH | −4 to 6 | 1 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 58 | 0 | 0 | 0 | 0 | 0 | 1 | 0 | 0 | 0 |
VKMDAEFRHD | −3 to 7 | 31 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 1 | 0 | 0 | 0 | 0 | 0 | 13 |
KMDAEFRHDS | −2 to 8 | 94 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 2 | 7 | 0 | 12 | 0 | 0 | 0 | 0 | 0 | 52 |
MDAEFRHDSG | −1 to 9 | 420 | 12 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 19 | 116 | 0 | 17 | 0 | 0 | 2 | 6 | 0 | 121 |
DAEFRHDSGY | 1–10 | 1983 | 1669 | 36 | 1721 | 3840 | 5193 | 2838 | 948 | 1675 | 1034 | 42,313 | 1284 | 274 | 81 | 1797 | 6024 | 4093 | 27,596 | 20,968 |
AEFRHDSGYE | 2–11 | 2 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 3 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
EFRHDSGYEV | 3–12 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
FRHDSGYEVH | 4–13 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
RHDSGYEVHH | 5–14 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
HDSGYEVHHQ | 6–15 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
DSGYEVHHQK | 7–16 | 214 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
SGYEVHHQKL | 8–17 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
GYEVHHQKLV | 9–18 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 16 | 0 | 0 | 0 |
YEVHHQKLVF | 10–19 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 10 | 0 | 0 | 0 |
EVHHQKLVFF | 11–20 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
VHHQKLVFFA | 12–21 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 27 | 0 | 0 | 0 |
HHQKLVFFAE | 13–22 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
HQKLVFFAED | 14–23 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
QKLVFFAEDV | 15–24 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |
DAEFRHDSGYEVHHQKLVFFAEDVGSNK | 1–28 | 685 | 161 | 220 | 295 | 450 | 715 | 1163 | 478 | 430 | 339 | 509 | 279 | 284 | 39 | 226 | 906 | 1157 | 893 | 1321 |
NOTE. The in vitro anti-Aβ antibody epitope mapping is a competitive binding inhibition enzyme-linked immunoassay for determination of binding residues of anti-Aβ antibody within the target region; the method is described in Section 2. The N-terminal Aβ1–10 (DAEFRHDSGY) peptide (given in bold) was identified to react most strongly with the serum samples collected on week 16 from each of the 19 patients immunized with UB-311; the results show 100% responder rate after immunization at weeks 0, 4, and 12. The numbers represent the dilution factor of each serum sample that corresponds to the 50% binding inhibition (IC50) by each of the 24 Aβ 10-mer peptides.