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. 2017 Jul 20;158(10):3212–3234. doi: 10.1210/en.2017-00468

Table 2.

Indicators of Enhancer Activation Are Specifically Enriched at NRFEs in Response to Hormone

Figure/Table ID Technology Comparing Motif Peak Selection Criteria Datasets
Hormone-regulated eRNA transcription
Fig. 4(a); Supplemental Table 3:1 Gro-Seq Veh vs E2 ERE B4 74
Fig. 4(b); Supplemental Table 3:3 Gro-Seq Veh vs DHT or Dex HRE B4 10
 Supplemental Table 3:2 Gro-Seq Veh vs E2 ERE B4–B20 74
 Supplemental Table 3:4 Gro-Seq Veh vs DHT or Dex HRE B4–B20 10
Hormone-regulated RNAPII occupancy
Fig. 4(c); Supplemental Table 3:5 RNAPII ChIP-Seq Veh vs E2 ERE D1000 8
Fig. 4(d); Supplemental Table 3:12 RNAPII ChIP-Seq Veh vs Cort, Dex, or Pred HRE D1000 3
 Supplemental Table 3:6 RNAPII ChIP-Seq Veh vs E2 ERE D1000–D20000 8
 Supplemental Table 3:7 RNAPII ChIP-Seq Veh vs E2 ERE L4–L20 8
 Supplemental Table 3:8 RNAPII ChIP-Seq: ERα-WT and ERα-KIKO Veh vs E2 ERE L4–L20 2
 Supplemental Table 3:9 RNAPII ChIP-Seq: ERα-WT and ERα-KIKO Veh vs E2 HRE L4–L20 2
 Supplemental Table 3:10 RNAPII ChIP-Seq Veh vs E2, Tam, or Fulv ERE L4–L10 3
 Supplemental Table 3:13 RNAPII ChIP-Seq Veh vs Cort, Dex, or Pred HRE D1000–D20000 3
Hormone-regulated recruitment of coregulators and chromatin remodeling proteins
Fig. 4(e); Supplemental Table 3:14 p300 ChIP-Seq Veh vs E2 ERE L4 2
Fig. 4(f); Supplemental Table 3:16 p300 ChIP-Seq Veh vs Dex, T, P4, or R5020 HRE L4 32
 Supplemental Table 3:15 p300 ChIP-Seq Veh vs E2 ERE L4–L20 2
 Supplemental Table 3:17 p300 ChIP-Seq Veh vs Dex, T, P4, or R5020 HRE L4–L20 32
Fig. 4(g); Supplemental Table 3:18 FoxA1 ChIP-Seq Veh vs E2 ERE L4 20
Fig. 4(h); Supplemental Table 3:20 FoxA1 ChIP-Seq Veh vs Dex, T, or R1881 HRE L4 10
 Supplemental Table 3:19 FoxA1 ChIP-Seq Veh vs E2 ERE L4–L20 20
 Supplemental Table 3:21 FoxA1 ChIP-Seq Veh vs Dex, T, or R1881 HRE L4–L20 10
 Supplemental Table 3:22 FoxA1 ChIP-Seq AR-C562S vs AR-WT HRE L4–L20 1
 Supplemental Table 3:23 FoxA1 ChIP-Seq AR-WT vs AR-Q640X HRE L4–L20 1
Fig. 4(i); Supplemental Table 3:24 DNase HSS ChIP-Seq Veh vs E2 ERE L4 12
Fig. 4(j); Supplemental Table 3:26 DNase HSS ChIP-Seq Veh vs Cort, Dex, or T HRE L4 20
 Supplemental Table 3:25 DNase HSS ChIP-Seq Veh vs E2 ERE L4–L20 12
 Supplemental Table 3:27 DNase HSS ChIP-Seq Veh vs Cort, Dex, or T HRE L4–L20 20
 Supplemental Table 3:28 Cohesin ChIP-Seq: STAG1 and RAD21 Veh vs E2 ERE L4–L20 2
 Supplemental Table 3:29 Cohesin ChIP-Seq: STAG1 and RAD21 CTCF-knockdown vs CTL ERE L4–L20 2
 Supplemental Table 3:30 PIAS1 ChIP-Seq Veh vs R1881 HRE L4–L20 2
 Supplemental Table 3:31 AR ChIP-Seq siPIAS1 vs CTL HRE L4–L20 2
 Supplemental Table 3:32 FoxA1 ChIP-Seq siPIAS1 vs CTL HRE L4–L20 2
 Supplemental Table 3:33 Sumo2/3 ChIP-Seq Veh vs R1881 HRE L4–L20 2
 Supplemental Table 3:34 Sumo2/3 ChIP-Seq GR-K721R vs GR-WT HRE L4–L20 2
 Supplemental Table 3:35 GR ChIP-Seq GR-K721R vs GR-WT HRE L4–L20 2
 Supplemental Table 3:36 GR ChIP-Seq siHic5 vs CTL HRE L4–L20 2
 Supplemental Table 3:37 HDAC 2 and 3 ChIP-Seq Veh vs DHT HRE L4–L15 2
 Supplemental Table 3:38 EZH2 ChIP-Seq Veh vs DHT HRE L4–L20 1
 Supplemental Table 3:39 TOP1 ChIP-Seq Veh vs DHT HRE L4–L10 1
 Supplemental Table 3:40 MRE11 ChIP-Seq Veh vs DHT HRE L4–L15 1
 Supplemental Table 3:41 Gro-Seq: Veh and DHT siTOP1 or siMRE11 vs CTL HRE B4–B20 8
Hormone-regulated transcription factor recruitment
 Supplemental Table 3:42 GATA3 ChIP-Seq Veh vs E2 ERE L4–L20 5
 Supplemental Table 3:43 GATA3 ChIP-Seq: Trans GATA3-WT vs GATA3-C318R or GATA3-N320K ERE L4–L20 2
 Supplemental Table 3:44 ERα ChIP-Seq siGATA3 vs CTL ERE L4–L20 1
 Supplemental Table 3:45 AR ChIP-Seq siGATA2 vs CTL HRE L4–L20 2
 Supplemental Table 3:46 RARα/γ ChIP-Seq Veh vs E2 ERE L4–L20 2
 Supplemental Table 3:47 RARα/γ ChIP-Seq: Trans RARα/γ-WT vs RARα/γ-pBox or RARα/γ-ZF ERE L4–L20 4
 Supplemental Table 3:48 Gro-Seq: Veh and E2 shRARs vs CTL ERE B4–B20 4
 Supplemental Table 3:49 p300 ChIP-Seq shRARs vs CTL ERE L4–L20 1
 Supplemental Table 3:50 ERα ChIP-Seq shRARs vs CTL ERE L4–L20 1
 Supplemental Table 3:51 pERα-S118 ChIP-Seq shRARs vs CTL ERE L4–L20 1
 Supplemental Table 3:52 Med1 ChIP-Seq Veh vs E2 ERE L4–L20 2
 Supplemental Table 3:53 Med1 ChIP-Seq: shCTL and shRARs Veh vs E2 ERE L4–L20 2
 Supplemental Table 3:54 Gro-Seq siSMC3 vs CTL ERE B4–B20 2
 Supplemental Table 3:55 AP2γ ChIP-Seq Veh vs E2 ERE L4–L20 1
 Supplemental Table 3:56 Gro-Seq: Veh and E2 shAP2γ vs CTL ERE B4–B20 4
 Supplemental Table 3:57 Stat3 ChIP-Seq Veh vs Dex HRE L4–L20 3
 Supplemental Table 3:58 ERG ChIP-Seq Veh vs DHT HRE L4–L20 1
 Supplemental Table 3:59 CEBP-β ChIP-Seq and ChIP-Exo Veh vs Dex or Pred HRE L4–L20 4
 Supplemental Table 3:60 CREB1 ChIP-Seq Veh vs Dex HRE L4–L20 2
 Supplemental Table 3:61 DNase HSS ChIP-Seq dn-CEBP-β vs CTL HRE L4–L20 2
 Supplemental Table 3:62 AP1 ChIP-Seq Veh vs Dex HRE L4–L10 1
 Supplemental Table 3:63 AP1 ChIP-Seq Veh vs Compound A HRE L4–L15 1
 Supplemental Table 3:64 Gro-Seq Veh vs Dex or Compound A HRE B4–B15 2

Summary of genomic features analyzed. See also Supplemental Tables 3:1–64.

Abbreviations: Cort, corticosterone; CTL, control; Dex, dexamethasone; DHT, 5α-dihydrotestosterone; dnCEBP-β, dominant negative-CEBP-β; Fulv, fulvestrant; HSS, hypersensitivity site; Pred, prednisolone; R1881, methyltrienolone; R5020, promegestone; shAP2γ, knockdown of AP2γ; shRAR, knockdown of RARα/γ; siGATA2, knockdown of GATA2; siGATA3, knockdown of GATA3; siHic5, knockdown of Hic5; siMRE11, knockdown of MRE11; siPIAS1, knockdown of PIAS1; siSMC3, knockdown of cohesin subunit SMC3; siTOP1, knockdown of TOP1; T, testosterone; Tam, tamoxifen; Veh, vehicle.