Figure 17.
(a) Comparison of experimentally verified HIV gp41 inhibitor NB-2 (gray box)101 to 12 members of a congeneric series of de novo designed compounds. The de novo molecule identifier, ZINC ID of the purchasable NB-2 analog, energy score, and pose classifier are listed for each compound. (b) This congeneric series adopted 3 related poses (labeled 1–3). HIV gp41 receptor shown as gray surface, key chelating Lys 29 residue shown as purple surface and sticks, de novo designed molecules shown as green sticks.