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. 2017 Oct 31;7:14453. doi: 10.1038/s41598-017-14776-0

Table 6.

In vitro Human liver microsomal stability data.

Compounds T1/2,int (min) CLint,app (µL/min/mg)
1a 10.20 169.81
1i 92.55 18.71
3a 53.29 32.50

CLint,app range: 14.4–577.5 µL/min/mg; T1/2,int range: 3–120 min; LM conc: 0.4 mg/mL.