Table 1.
Hit ID | Structure | Pseudovirus
|
Infectious EBOV
|
||||
---|---|---|---|---|---|---|---|
IC50, μM
|
CC50, μM | IC50, μM | CC50, μM | SI | |||
EBOV | MARV | ||||||
cp3 | 6.9 ± 1.4 | 9.1 ± 1.0 | 156.9 ± 12.5 | 5.2 ± 0.7 | 223 | 43 | |
cp5 | 4.1 ± 1.3 | 9.0 ± 1.8 | >264.3 | 4.0 ± 0.6 | 264 | 66 | |
cp11 | 3.8 ± 0.7 | 5.6 ± 0.7 | 74.9 ± 19.4 | 7.5 ± 1.3 | 85 | 11 | |
cp13 | 6.4 ± 0.9 | 9.2 ± 1.7 | >291.2 | 8.7 ± 0.9 | 150 | 17 | |
cp15 | 1.8 ± 0.7 | 5.1 ± 1.6 | 50.3 ± 2.7 | 5.2 ± 0.2 | 80 | 16 | |
cp16 | 3.8 ± 0.9 | 6.9 ± 0.9 | 77.8 ± 14.0 | 5.1 ± 0.1 | 146 | 28 | |
cp19 | 2.4 ± 0.3 | 4.8 ± 0.4 | 48.0 ± 4.3 | 3.7 ± 1.5 | 71 | 19 |
Abbreviations: CC50, 50% cytotoxic concentration; EBOV, Ebolavirus; IC50, 50% inhibitory concentration; MARV, Marburgvirus; SI, selectivity index. Data are means ± SD from at least two independent experiments.