| 5-FU | 5-Fluorouracil |
| ABC | ATP-Binding Cassette |
| AGT | O6-alkylguanine transferase |
| Ahr | Aryl hydrocarbon receptor |
| ALAS1 | Aminolevulinic acid synthase |
| ASPS | Advanced sleep phase syndrome |
| ATM | Ataxia telangiectasia mutated |
| BAX | BCL-2-associated X protein |
| BMAL1 | Brain and muscle aryl hydrocarbon receptor nuclear translocator 1 |
| CAR | Constitutive androstan receptor |
| CCGs | Clock controlled genes |
| CDC2 | Cyclin-dependent kinase 2 |
| CES | Carboxylesterase |
| ChronoDDS | Chrono-drug delivery system |
| ChronoPD | Chronopharmacodynamics |
| ChronoPK | Chronopharmacokinetics |
| CKIε | Casein kinase Iε |
| CLOCK | Circadian locomotor output cycles kaput |
| Cmax | Maximum plasma concentration |
| Cry | Cryptochrome |
| CTS | Circadian timing system |
| Cyc | Cyclin |
| CYCLOPS | Cyclic ordering by periodic structure |
| CYP450 | Cytochrome P-450 |
| DBP | Albumin D-site-binding protein |
| DDS | Drug delivery systems |
| DPYD | Dihydropyrimidine dehydrogenase |
| DSPS | Delayed sleep phase syndrome |
| EGFR | Epidermal growth factor receptor |
| ERK/MAPK | Extracellular signal-regulated kinase/mitogen-activated protein kinase |
| FASPS | Familial advanced sleep phase syndrome |
| GSH | Reduced glutathione |
| GST | Glutathione-S-transferases |
| HLF | Hepatic leukemia factor |
| Hsd3b | 3β-hydroxysteroid dehydrogenase |
| IFN-β | Interferon-β |
| ISGF | Interferon-stimulated gene factor |
| MDR1 | Multidrug resistance protein 1 (ABCB1, P-glycoprotein, P-gp in human) |
| Mdr1 | Multidrug resistance protein 1 (abcb1a/b mdr1a/b, P-gp in rodents) |
| MR | Modified Release |
| Mrp | Multidrug resistance-associated protein (Abcc) |
| mTOR | Mammalian target of rapamycin |
| NAT | N-acetyl transferases |
| NFIL3/E4BP4 | Nuclear factor, interleukin 3 regulated |
| NPAS2 | Neuronal PAS-domain protein 2 |
| Oatp | Organic anion transporter polypeptide |
| Oct | Organic cation transporter |
| Octn1 | Oct novel type 1 |
| p21WAF1 | p21 wild-type p53 fragment 1 |
| PARbZip | Proline-acidic amino acid-rich basic leucine zipper |
| PD | Pharmacodynamics |
| PDGF | Platelet-derived growth factor |
| Per | Period |
| P-gp | P-glycoprotein |
| PI3K/AKT | Phosphatidylinositol-3-kinase/protein kinase B |
| PK | Pharmacokinetics |
| POR | P450 oxidoreductase |
| PPAR-α | Peroxisome proliferator activated receptor-alpha |
| PTX | Paclitaxel |
| PTX-NPs | PTX-loaded polymeric nanoparticles |
| PXR | Pregnane X receptor |
| REV-ERB/NR1D | Reverse strand of ERB |
| RORs | Retinoic acid-receptor-related orphan receptor |
| SCN | Suprachiasmatic nuclei |
| SLC | Solute carrier |
| SULT | Sulfotransferases |
| TEF | Thyrotroph embryonic factor |
| Top1 | Topoisomerase 1 |
| TS | Thymidylate synthase |
| UDP | Uridine diphosphate |
| UGT | Glucuronosyl transferase |
| VEGF | Vascular endothelial growth factor |
| WBC | White blood cells |