Table 1.
Strain | Genotype | Letermovir |
||||
---|---|---|---|---|---|---|
EC501 | SD2 | N3 | Fold4 | Δ5 | ||
Control Strains | ||||||
4190 | WT UL56 Frt | 3.7 | 0.77 | 79 | ||
4272 | WT UL89 Frt | 3.5 | 0.65 | 26 | ||
4194 | UL56 V231L | 21 | 3.4 | 81 | 5.6 | |
4296 | UL56 V236M | 115 | 13 | 11 | 32 | |
4192 | UL56 L241P | 633 | 136 | 25 | 173 | |
4315 | UL56 R369M | 60 | 8.6 | 20 | 16 | |
4274 | UL89 D344E | 5.5 | 1.1 | 24 | 1.6 | |
Newly Phenotyped Mutants | ||||||
4244 | UL56 S229F | 6.6 | 1.1 | 11 | 1.8 | |
4324 | UL56 S229F L254F L257I | 198 | 25 | 12 | 54 | |
4292 | UL56 L254F | 12 | 2.1 | 10 | 3.2 | |
4346 | UL56 L257F | 31 | 6.1 | 10 | 8.6 | |
4312 | UL56 N368D | 7.4 | 1.5 | 10 | 2.0 | |
4317 | UL51 P91S | 7.6 | 1.7 | 43 | 2.1 | |
4318 | UL51 P91S UL56 S229F | 23 | 3.3 | 10 | 6.3 | 3.5 |
4348 | UL51 P91S UL56 S229F L254F L257I | 1060 | 137 | 12 | 290 | 5.4 |
4319 | UL51 P91S UL56 V236M | 101 | 10 | 10 | 28 | 0.9 |
4325 | UL51 P91S UL56 R369M | 460 | 53 | 10 | 126 | 7.7 |
4400 | UL51 P91S UL89 D344E | 14 | 1.2 | 17 | 4.0 | 2.6 |
Mean letermovir EC50 in nM
Standard deviation of EC50 values
Number of replicates (performed on at least 4 separate dates)
Ratio of EC50 value to that of wild type control strain (values >1.5 in bold)
Fold change in EC50 value resulting from addition of UL51 P91S to UL56 or UL89 mutation