Table 3.
Compound | n | m | Diamine | X |
---|---|---|---|---|
27 | 1 | 2 | Homopiperazine | H |
28 | 1 | 1 | Piperazine | H |
29 | 0 | 2 | Homopiperazine | 4-OMe |
30 | 1 | 2 | Homopiperazine | 4-OMe |
31 | 1 | 1 | Piperazine | 4-OMe |
32 | 0 | 1 | Piperazine | 4-OMe |
33 | 0 | 2 | Homopiperazine | 3,5-(OMe)2 |
34 | 1 | 1 | Piperazine | 3,5-(OMe)2 |
35 | 1 | 1 | Piperazine | 3,5-(OMe)2 |
36 | 1 | 2 | Homopiperazine | 4-F |
37 | 1 | 1 | Piperazine | 4-F |