Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.
Activity towards the calcium mobilizing response in GPR103-transfected cells of different 26FRa analogues.
| entry | pseudopeptides | EC50 (nM) |
| 1 | Gly-Gly-Phe-Ser-Phe-Arg-Phe-NH2 | (739 ± 149) |
| 2 | Gly-ψ[(Z)-CF=CH]-Gly-Phe-Ser-Phe-Arg-Phe-NH2 | (618 ± 104) |
| 3 | Gly-ψ[(E)-CF=CH]-Gly-Phe-Ser-Phe-Arg-Phe-NH2 | (538 ± 13) |
| 4 | Gly-Gly-ψ[(Z)-CF=CH]-D-Phe-Ser-Phe-Arg-Phe-NH2 | 6752 |
| 5 | Gly-Gly-ψ[(Z)-CF=CH]-L-Phe-Ser-Phe-Arg-Phe-NH2 | (1720 ± 1010) |
