Table 1.
Pax2 Specific Inhibitors Identified by Virtual Screening
| PRS4-LUC | CMV-LUC | ||
|---|---|---|---|
| Structure | CCG ID | IC50 (µM) | IC50 (µM) |
|
3036 | 106.7 ± 11.3 | >500 |
|
3647 | 126.5 ± 26.5 | >500 |
|
21766 | 126.4 ± 19.8 | >500 |
|
21767 | 51.9 ± 4.9 | >500 |
|
100613 | 48.6 ± 6.5 | 291.3 ± 75.6 |