Table 4. Structures and experimental activity of novel inhibitors targeting menin–MLL interaction.
| Inhibitor | Structure | IC50 [μM] |
| 1 |
|
0.193 |
| 2 |
|
0.65 |
| 3 |
|
1.30 |
| 4 |
|
1.40 |
| 5 |
|
2.00 |
| 6 |
|
20.00 |
| 7 |
|
200.00 |
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