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. 2017 Sep 14;39(2):243–250. doi: 10.1038/aps.2017.96

Table 1. The kinase panel screening data of SOMCL-085.

Kinase IC50 (nmol/L)a
FGFR1 1.8±0.2
FGFR2 1.9±0.4
FGFR3 6.9±1.2
FGFR4 319.9±24.9
VEGFR-1 5.6±0.5
VEGFR-2 1.2±0.2
PDGFR-α 22.6±10.5
PDGFR-β 7.8±1.8
EGFR >1000
ErbB2 >1000
ErbB4 >1000
ABL >1000
c-Src >1000
EPH-A2 >1000
IGF1R >1000
ALK >1000
LTK >1000
ROS1 >1000
c-Met >1000
AXL >1000

aValues are the mean±SD of two independent assays.