Table 1. The kinase panel screening data of SOMCL-085.
| Kinase | IC50 (nmol/L)a |
|---|---|
| FGFR1 | 1.8±0.2 |
| FGFR2 | 1.9±0.4 |
| FGFR3 | 6.9±1.2 |
| FGFR4 | 319.9±24.9 |
| VEGFR-1 | 5.6±0.5 |
| VEGFR-2 | 1.2±0.2 |
| PDGFR-α | 22.6±10.5 |
| PDGFR-β | 7.8±1.8 |
| EGFR | >1000 |
| ErbB2 | >1000 |
| ErbB4 | >1000 |
| ABL | >1000 |
| c-Src | >1000 |
| EPH-A2 | >1000 |
| IGF1R | >1000 |
| ALK | >1000 |
| LTK | >1000 |
| ROS1 | >1000 |
| c-Met | >1000 |
| AXL | >1000 |
aValues are the mean±SD of two independent assays.