Table 1.
Experiment 1
|
Experiment 2
|
Experiment 3
|
Average IC50 ratios | ||||
---|---|---|---|---|---|---|---|
IC50 (nM) | IC50 ratio | IC50 (nM) | IC50 ratio | IC50 (nM) | IC50 ratio | ||
Tamoxifen | 106 | 1 | 88 | 1 | 188 | 1 | 1 |
N-desmethyltamoxifen | 189 | 0.56 | 573 | 0.15 | 430 | 0.44 | 0.38 |
(Z)-4-hydroxytamoxifen | 18 | 5.89 | 7 | 12.6 | 4 | 47 | 21.8 |
(Z)-Endoxifen | 8 | 13.3 | 4 | 22 | 1 | 188 | 74.4 |
IC50 = half maximal inhibitory concentration