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. Author manuscript; available in PMC: 2018 Feb 19.
Published in final edited form as: Brain Res Bull. 2016 Apr 29;126(Pt 1):111–126. doi: 10.1016/j.brainresbull.2016.04.011

Table 1.

Effect of pyrrolidinophenones on inhibition of synaptosomal monoamine transporters (Marusich et al., 2014); see Table 2 for chemical structures.

IC50 (nM)

DAT NET SERT
MDPV 4.1 25.9 3,305
α-PVP 12.8 14.2 >10,000
α-PBP 63.3 91.5 >10,000
α-PPP 196.7 444.7 >10,000