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. Author manuscript; available in PMC: 2019 Mar 1.
Published in final edited form as: J Neural Transm (Vienna). 2017 Aug 31;125(3):337–363. doi: 10.1007/s00702-017-1774-z

Table 1.

Species Age Sex PD patients/MPTP dose MPTP regimen Parkinsonian clinical symptom Pathology observation (Nigral dopamine cell/striatal DA levels loss in %) Reference
Midbrain dopaminergic neurons
Human 62–83 M,F PD Fully Parkinsonian VM – 71
VL - 91
PL – 61
DM – 47
DL - 57
(Fearnley and Lees 1991)
Human 72 ± 4 PD Fully Parkinsonian SNC v nigrosomes – 95
SNC v matrix - 80
SNC d - 57
(Damier et al. 1999b;
Damier et al. 1999d)
Callithrix jacchus F 1–4 mg/kg/day for 5 days,i.p Acute high dose treatment Fully Parkinsonian SNC 82
VTA 59
(Waters et al. 1987)
Papio papio 0.2–0.5 mg/kg i.v once a week until a full parkinsonian Chronic low dose treatment Fully Parkinsonian VM - 73.8
VL - 90.9
PL - 89.5
DM – 46
DL - 56.6
VTA - 53
(Varastet et al. 1994)
Cercopithec us aethiops 4 – 6 M 0.4 – 0.6 mg/kg i.m Progressive intoxication: (injections spaced 4 to 5 days) Chronic low/high dose treatment Fully Parkinsonian monkeys SNC - 71
RRF - 35
VTA - 34
(Mounayar et al. 2007)
Macaca mulatta 8–9 Young
15–17 Middle
21–31 Old
F 2.3–3.00 mg, unilateral intracarotid administration Single dose Hemiparkinsonia monkey SNC - 81.8
SNC - 82.8
SNC-81.0
(Collier et al. 2007)
Macaca mulatta 3–6 F 0.2–0.5 mg/kg i.m once a week until a full parkinsonian Chronic low dose treatment Moderate Parkinsonian monkeys
Fully Parkinsonian monkeys
SNC v - 64
SNC d - 53
VTA – 42

SNC v - 85
SNC d - 73
VTA – 60
(Masilamoni et al. 2011b)
Macaca fascicularis 4–5 M 0.5 mg/kg i.v once in 2 weeks Chronic low dose treatment Moderate Parkinsonian monkeys
Fully Parkinsonian monkeys
SNC - 74
RRF - 40
VTA – 34

SNC - 84
RRF - 45
VTA - 33
(Blesa et al. 2012)
Nigrostriatal Dopamine Innervation
Human - - Fully Parkinsonian Pre-commissural CA-90
Commissural CA - 82
Post-commissural CA- 70
Pre-commissural PU-93
Commissural PU – 97
Post-commissural PU-98
(Kish et al. 1988)
Human Fully Parkinsonian CA-84
PU-98
(Pifl et al. 1988b)
Human Fully Parkinsonian CA-80
PU-98
(Kish et al. 2008)
Macaca mulatta 10–17 0.15 mg/kg for the first 3 days and consecutively 0.24 – 0.4 mg/kg per day until severe Parkinson-like symptoms Acute low dose treatment Fully Parkinsonian monkeys CA-99
PU-99
(Pifl et al. 1988b)
Cercopithec us- aethiops subueus 0.4mg/kg for 5 days Acute low dose treatment Fully Parkinsonian monkeys CA 98
PU 96
(Elsworth et al. 1989)
Callithrix jaccus 1–2Y M,F 1.25–2.5 mg/kg s.c. was given twice a week up to development of symptom Chronic high dose treatment Fully Parkinsonian monkeys CA 95
PU 95
(Perez-Otano et al. 1991)
Macaca fascicularis daily injections (0.25–0.50 mg/kg) Acute low dose treatment Fully Parkinsonian monkeys PU 97
CA 98
(Alexander et al. 1992)
Macaca fascicularis 3 consecutive i.v injection at 0.7mg/day Acute high dose treatment Fully Parkinsonian monkeys CA 94 PU 93 (Hantraye et al. 1992)
Pupio pupio 0.4–0.6 mg/kg i.v once a week until a full parkinsonian Chronic low dose treatment Fully Parkinsonian monkeys CA 70
PU 90
(Hantraye et al. 1993)
Saimiri sciureus M,F single subcutaneous injection of 2 mg/kg MPTP
received multiple subcutaneous injections
Single dose
Acute intoxication
no behavioral signs of parkinsonism
Fully Parkinsonian monkeys
CA 63
PU 70
CA 95
PU 99
(Di Monte et al. 2000)
Cercopithec us- aethiops sabaeus 0.4mg/kg for 5 days Acute low dose treatment Asymptomatic
Mild
Moderate
Severe
CA 70; PU 58
CA 90; PU 68
CA 94; PU 92
CA99; PU 99
(Elsworth et al. 2000)
Caca fascicularis 3.1 ± 0.3 F 0.2 mg/kg, i.v. daily after 6 injections; D6 after 15 injections; D15 after 15 injections; D25 Acute low dose treatment Pre-symptomatic Appearance of symp.
Fully Parkinsonian monkeys
Loss of dopamine CA 50; PU 40
PU 85%; CA 90
CA 95; PU 95%
(Bezard et al. 2001)
Mucucu fusciculuris M Intracarotid injections
Single dose of 1.25 mg
Single dose of 2.5 mg
Acute low dose treatment hemiparkinsonism ipsilateral DA loss CA 99.4; PU, 99.8; AC 74.2
CA 99.3; PU 99.5; AC 90.1
(Guttman et al. 1990)
Macaca fascicularis 2–4 5–15 injections of 0.5–1.0 mg/kg spaced one week apart Chronic high dose treatment Fully Parkinsonian Pre-commissural CA-98
Commissural CA - 94
Post-commissural CA- 90
Pre-commissural PU-98
Commissural PU – 99
Post-commissural PU-99
(Perez-Otano et al. 1994a)
Macaca mulatta 3–6 F 0.2–0.5 mg/kg i.m once a week until full parkinsonian Chronic low dose treatment Moderate Parkinsonian monkeys
Fully Parkinsonian monkeys
CA - 63
PU - 80
CA - 80
PU - 90
(Masilamoni et al. 2011b)
Macaca fascicularis 4–5 M 0.5 mg/kg i.v once in 2 weeks Chronic low dose treatment Moderate Parkinsonian monkeys
Fully Parkinsonian monkeys
CA - 78
PU - 79
CA - 84
PU - 83
(Blesa et al. 2012)

VM – Ventral medial, VL - Ventral lateral, PL – Pars lateralis, DM – Dorsal medial part, DL - lateral part, CA- Caudate, PU- Putamen, SNC - Substantial nigra, SNC v- ventral, SNC-d-dorsal, VTA – Ventral tegmental area, RRF – Retrorubral area