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. 2016 May 5;1:8. doi: 10.1186/s41181-016-0013-5

Table 2.

Tumor-to-background ratios at different time points after injection of 44Sc/68Ga-labeled DOTA-RGD and NODAGA-RGD

44Sc-DOTA-RGD 68Ga-DOTA-RGD
U87MG 30 min p.i. 2 h p.i. 5 h p.i. 30 min p.i. 2 h p.i.
Tumor-to-blood 4.82 ± 1.60 40.1 ± 15.6 47.2 ± 18.0 4.34 ± 0.57 28.0 ± 4.26
Tumor-to-liver 0.99 ± 0.14 0.61 ± 0.04 2.90 ± 0.38 0.55 ± 0.09 0.48 ± 0.07
Tumor-to-kidney 1.16 ± 0.29 1.77 ± 0.13 1.82 ± 0.21 0.88 ± 0.07 1.74 ± 0.19
44Sc-NODAGA-RGD 68Ga-NODAGA-RGD
U87MG 30 min p.i. 2 h p.i. 5 h p.i. 30 min p.i. 2 h p.i.
Tumor-to-blood 4.73 ± 1.24 34.1 ± 7.62 30.5 ± 9.93 4.17 ± 0.47 114 ± 35.0
Tumor-to-liver 3.02 ± 0.40 3.01 ± 0.13 2.82 ± 0.21 1.72 ± 0.16 1.50 ± 0.20
Tumor-to-kidney 1.18 ± 0.28 2.68 ± 0.14 2.58 ± 0.24 0.89 ± 0.03 1.49 ± 0.21