Table 1.
Caco-2 Permeability
Compound | A ->B Papp (10-6 cm•s-1) | B ->A Papp (10-6 cm•s-1) | RE |
---|---|---|---|
Ranitidine | 0.2 | 1.3 | 8.1 |
Warfarin | 35.5 | 8.6 | 0.2 |
Talinolol | 0.3 | 5.4 | 16.8 |
38 | 1.1 | 20.3 | 18.2 |
38D-16 | 0.9 | 3.0 | 3.3 |
38D-21 | 2.7 | 7.0 | 2.6 |
38D-22 | 10.0 | 30.5 | 3.0 |
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