Table 3.
Screening of molecules on cardiac MMP-2 with gelatin zymography.
Code | Inhibition (%)±SEM at 100 μM final MMP inhibitor concentration |
---|---|
MMPI-1133 | 11.14 ± 1.58 |
MMPI-1140 | 81.08 ± 3.88 |
MMPI-1154 | 100 |
MMPI-1155 | 46.95 ± 19.06 |
MMPI-1157 | 100 |
MMPI-1245 | 100 |
MMPI-1247 | 100 |
MMPI-1248 | 100 |
MMPI-1252 | 100 |
MMPI-1253 | 100 |
MMPI-1254 | 100 |
MMPI-1260 | 100 |