. 2018 Feb 13;9(4):354–358. doi: 10.1021/acsmedchemlett.7b00546

Table 1. Activity and Selectivity of HTS Hit and Close-in Analogues^a.

graphic file with name ml-2017-00546m_0005.jpg

#	R	FSK AC₄₀ (μM)	CV AC₄₀ (μM)	SSK AC₄₀ (μM)
1	S-Me	7	>49	>39
2	R-Me	>49
3	H	>49

FSK = fast skeletal muscle; CV = cardiac muscle; SSK = slow skeletal muscle.

Table 1. Activity and Selectivity of HTS Hit and Close-in Analoguesa.