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. 2018 Mar 26;9(4):312–317. doi: 10.1021/acsmedchemlett.7b00487

Table 2. Pharmacokinetic Profiles of Compound 10 in Sprague–Dawley Ratsa.

compds Cmax (ng/mL) Tmax (h) T1/2 (h) AUC(0-inf) (ng/mL·h) F (%)
2 (Po) 5560 ± 967 0.8 4.5 ± 0.8 30747 ± 785  
10 (Po) 5765 ± 1276 2.0 3.4 ± 0.1 33534 ± 225 18
10 (Iv) 12039 ± 1762 0.083 1.4 ± 0.05 3646 ± 201  
a

Data are presented as mean ± SD.