Table 2.
Commonly used commercially available oxytocin (OT) and arginine-vasopressin (AVP) receptor agonists and antagonists.
Category | Compound | Name/acronym | Supplier |
---|---|---|---|
OTR agonist | [Thr4, Gly7]-OT | TGOT | Abgent; Bachem |
WAY267, 464*# | N/A | Tocris | |
OTR antagonist | d(CH2)5-Tyr(Me)-[Orn8]-vasotocin | N/A | Bachem |
V1aR antagonist | d(CH2)5[Try(Me)2]AVP | Manning Compound | Sigma-Aldrich |
SR49059* | N/A | Tocris; Sigma-Aldrich | |
V1bR antagonist | SSR149415* | Nelivaptan | Sigma-Aldrich |
indicates non-peptide agonists/antagonists.
is also a V1aR antagonist [126].