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Chemical starting points profiled in the NAK family assay panel
| Cmpd | Binding displacement assay Ki (μM) | NAK selectivityb | |||
|---|---|---|---|---|---|
| GAK | AAK1 | BMP2K | STK16 | ||
| 1 | 0.0039 | 54 | >100 | 17 | 4300 |
| 2 | 0.0015 | 2.8 | 8.6 | >10 | 1900 |
| 3 | 0.015 | 3.1 | 6.6 | >10 | 210 |
Selectivity against the nearest NAK family member
