Table 5. . Kd (nM) determined via DiscoverX Kd Elect service.
| Kinase | HSN286 | HSN356 |
|---|---|---|
| AURKA | >30,000 | 5100 |
| BLK | 3.9 | 1.2 |
| CDK6 | 28,000 | ND |
| CDK9 | 2300 | ND |
| FAK | 5100 | 4700 |
| FGR | 7 | 7.9 |
| FLT3 | 7.2 | 1.3 |
| FYN | 28 | 38 |
| HCK | 3.6 | 2.5 |
| KIT | 42 | 7.2 |
| LYN | 11 | 5.4 |
| PIK3CA | 26,000 | >30,000 |
| PIM1 | 11,000 | 19,000 |
| PLK1 | >30,000 | 9600 |
| SRC | 16 | 15 |
ND: Not determined.