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. 2017 May 11;9(11):1213–1225. doi: 10.4155/fmc-2017-0067

Table 5. . Kd (nM) determined via DiscoverX Kd Elect service.

Kinase HSN286 HSN356
AURKA >30,000 5100

BLK 3.9 1.2

CDK6 28,000 ND

CDK9 2300 ND

FAK 5100 4700

FGR 7 7.9

FLT3 7.2 1.3

FYN 28 38

HCK 3.6 2.5

KIT 42 7.2

LYN 11 5.4

PIK3CA 26,000 >30,000

PIM1 11,000 19,000

PLK1 >30,000 9600

SRC 16 15

ND: Not determined.