Table 4. PTD2 biochemical IC50 values for a panel of HMT enzymes.
| Enzyme | Biochemical IC50 (μM) |
|---|---|
| WHSC1 941–1240 | 22 ± 2 |
| WHSC1L1 1054–1285 | 3.2 ± 0.2 |
| EZH1 | >200 |
| EZH2 | >200 |
| G9a | >200 |
| SMYD2 | >200 |
| SETDB1 | >200 |
| PRMT6 | >200 |
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