Table 2. Pharmacokinetic parameters after single intravenous bolus administration of SNF472 into rats.
1 mg/kg | 5 mg/kg | 10 mg/kg | |
---|---|---|---|
C0 (ng/mL) | 36775 | 84561 | 156750 |
t1/2 (min) | 1.8 | 6.6 | 7.8 |
AUC(0→t) (ng·h/mL) | 3491 | 19234 | 38752 |
MRT (0→∞) (h) | 1.65 | 0.33 | 0.19 |
Vz (L/kg) | 0.01 | 0.04 | 0.05 |
Cl (L/h/kg) | 0.29 | 0.26 | 0.26 |
C0: extrapolated concentration at time = 0 min; t1/2: half-life; AUC: area under the curve; MRT: mean residence time; Vz: volume of distribution; Cl: clearance